Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 16 hits in this display   

Target5-hydroxytryptamine receptor 4(GUINEA PIG)TBA
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  0.741nMAssay Description:Compound was tested for binding affinity against 5-HT4 receptor in guinea pig striata using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 4(GUINEA PIG)TBA
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  0.790nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)TBA
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  0.790nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInner capsid protein sigma-2(Reovirus type 1 (strain Lang) (T1L) (Mammalian ort...)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  15.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter capsid protein sigma-1(Mammalian orthoreovirus 3 Dearing)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  158nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  398nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  794nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Xenopus tropicalis)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed