Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 15 hits in this display
BDBM50079362(CHEMBL3417009 | US9663465, 9)
BDBM50079362(CHEMBL3417009 | US9663465, 9)
Ki: 6.60nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
BDBM50079362(CHEMBL3417009 | US9663465, 9)
BDBM50079362(CHEMBL3417009 | US9663465, 9)
BDBM50079362(CHEMBL3417009 | US9663465, 9)
BDBM50079362(CHEMBL3417009 | US9663465, 9)
BDBM50079362(CHEMBL3417009 | US9663465, 9)
BDBM50079362(CHEMBL3417009 | US9663465, 9)
Ki: 51nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in human Jurkat cell membranes after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
BDBM50079362(CHEMBL3417009 | US9663465, 9)
BDBM50079362(CHEMBL3417009 | US9663465, 9)
IC50: 16nMAssay Description:Inhibition of human erythrocyte AChE pre-incubated for 5 mins before acetylthiocholine iodide substrate by Ellman' methodMore data for this Ligand-Target Pair
BDBM50079362(CHEMBL3417009 | US9663465, 9)
BDBM50079362(CHEMBL3417009 | US9663465, 9)
BDBM50079362(CHEMBL3417009 | US9663465, 9)
BDBM50079362(CHEMBL3417009 | US9663465, 9)
IC50: 3.53E+3nMAssay Description:Inhibition of equine serum BuChE pre-incubated for 5 mins before butyrylthiocholine iodide substrate by Ellman' methodMore data for this Ligand-Target Pair
BDBM50079362(CHEMBL3417009 | US9663465, 9)