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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50390658(CHEMBL2070003)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of recombinant AKR1C3 using S-tetralol as substrate by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50390658(CHEMBL2070003)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of recombinant AKR1C3 using 1-acenaphthenol as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C2(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50390658(CHEMBL2070003)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of recombinant AKR1C2 using S-tetralol as substrate by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50390658(CHEMBL2070003)
Affinity DataIC50:  5.09E+4nMAssay Description:Inhibition of recombinant AKR1C4 using S-tetralol as substrate by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50390658(CHEMBL2070003)
Affinity DataIC50:  8.63E+4nMAssay Description:Inhibition of recombinant AKR1C1 using S-tetralol as substrate by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed