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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by
PubChem BioAssay
Ligand
BDBM55082
(N-[4-[(2-chlorobenzoyl)amino]-3-methoxy-phenyl]pic...)
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Affinity Data
EC50: 95.3nM
Assay Description:
Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University The primary pathophysiological change giving rise to the symptoms...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
PCBioAssay
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Target
Metabotropic glutamate receptor 4 [Q124R]
(Rattus norvegicus)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by
PubChem BioAssay
Ligand
BDBM55082
(N-[4-[(2-chlorobenzoyl)amino]-3-methoxy-phenyl]pic...)
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Copy InChI
Affinity Data
EC50: 110nM
Assay Description:
Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University The primary pathophysiological change giving rise to the symptoms...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
PCBioAssay
Copy BDB DOI
Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Vanderbilt University
Curated by
ChEMBL
Ligand
BDBM55082
(N-[4-[(2-chlorobenzoyl)amino]-3-methoxy-phenyl]pic...)
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Copy InChI
Affinity Data
EC50: 34nM
Assay Description:
Positive allosteric modulation of rat mGlu4 receptor expressed in HEK293 cells coexpressing GIRK assessed as thallium influx in presence of EC20 glut...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Vanderbilt University
Curated by
ChEMBL
Ligand
BDBM55082
(N-[4-[(2-chlorobenzoyl)amino]-3-methoxy-phenyl]pic...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 106nM
Assay Description:
Positive allosteric modulation of rat mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by
PubChem BioAssay
Ligand
BDBM55082
(N-[4-[(2-chlorobenzoyl)amino]-3-methoxy-phenyl]pic...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 99.5nM
Assay Description:
Positive allosteric modulation of human mGluR4 expressed in CHO cells coexpressing Gqi5 assessed as calcium mobilization
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI