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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
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kcal/mol
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Found
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Target
Serine/threonine-protein kinase B-raf [V600E]
(Homo sapiens (Human))
Cancer Research Uk Centre For Cancer Therapeutics
Ligand
BDBM25566
((4-{6-[(3,4,5-trimethoxyphenyl)amino]pyrazin-2-yl}...)
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Affinity Data
IC50: 2.60E+4nM
pH: 7.2 T: 2°C
Assay Description:
BRAF kinase activity was quantified using a DELFIA-based MEK1 phosphorylation assay. IC50 values were derived from the sigmoidal dose-response curves...
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