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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Platelet-derived growth factor receptor alpha
(Homo sapiens (Human))
National University Of Ireland
Curated by
ChEMBL
Ligand
BDBM50336466
((3S,5R,E)-5-chloro-16-hydroxy-14-methoxy-3-methyl-...)
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Affinity Data
IC50: 1.20E+3nM
Assay Description:
Inhibition of human recombinant PDGFRalpha in cell free system after 60 mins
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
National University Of Ireland
Curated by
ChEMBL
Ligand
BDBM50336466
((3S,5R,E)-5-chloro-16-hydroxy-14-methoxy-3-methyl-...)
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Affinity Data
IC50: 3.40E+4nM
Assay Description:
Inhibition of human recombinant FLT-3 kinase expressed in insect cells after 90 mins
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Vascular endothelial growth factor receptor 3
(Homo sapiens (Human))
National University Of Ireland
Curated by
ChEMBL
Ligand
BDBM50336466
((3S,5R,E)-5-chloro-16-hydroxy-14-methoxy-3-methyl-...)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of human recombinant VEGFR3 in cell free system after 90 mins
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
National University Of Ireland
Curated by
ChEMBL
Ligand
BDBM50336466
((3S,5R,E)-5-chloro-16-hydroxy-14-methoxy-3-methyl-...)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of human recombinant c-kit kinase in cell free system after 30 mins
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI