Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBifunctional protein GlmU(Escherichia coli)
Csir-Indian Institute Of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50075339(CHEMBL3414910)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Streptococcus pneumoniae)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50365079(CHEMBL1951168)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Streptococcus pneumoniae acetyltransferase activity of GlmU using acetyl-CoA and glucosamine-1-phosphate after 30 mins by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Csir-Indian Institute Of Integrative Medicine

Curated by ChEMBL
LigandPNGBDBM50075339(CHEMBL3414910)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed