Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Avanti Biosciences

Curated by ChEMBL
LigandPNGBDBM50296234((-)-epigallocatechin-3-(3''-O-methyl)gallate | (2R...)
Affinity DataIC50:  429nMAssay Description:Inhibition of DYRK1A (unknown origin) using HT-497 as substrate preincubated with compound followed by substrate addition and measured after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296234((-)-epigallocatechin-3-(3''-O-methyl)gallate | (2R...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296234((-)-epigallocatechin-3-(3''-O-methyl)gallate | (2R...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296234((-)-epigallocatechin-3-(3''-O-methyl)gallate | (2R...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed