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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
ALK tyrosine kinase receptor
(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50185286
(CHEMBL3823256)
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Affinity Data
IC50: 0.330nM
Assay Description:
Inhibition of human ALK using poly[Glu:Tyr] (4:1) as substrate and [gamma-33P]ATP measured after 1 hr
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Insulin-like growth factor 1 receptor
(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50185286
(CHEMBL3823256)
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Copy InChI
Affinity Data
IC50: 0.400nM
Assay Description:
Inhibition of human IGF1R using KKKSPGEYVNIEFG as substrate and [gamma-33P]ATP measured after 1 hr
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Insulin receptor
(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50185286
(CHEMBL3823256)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.70nM
Assay Description:
Inhibition of human InsR using myelin basic protein as substrate and [gamma-33P]ATP measured after 1 hr
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI