Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM135949(US8853203, 3 | US8853203, 8 | US9650377, Example 8)
BDBM135949(US8853203, 3 | US8853203, 8 | US9650377, Example 8)
BDBM135949(US8853203, 3 | US8853203, 8 | US9650377, Example 8)
IC50: 220nMAssay Description:Activity of compounds of the present invention was examined by determination to what extent the glutamate-induced elevation of the intracellular calc...More data for this Ligand-Target Pair
BDBM135949(US8853203, 3 | US8853203, 8 | US9650377, Example 8)
IC50: 220nMAssay Description:Activity of compounds of the present invention with respect to mGluR1 antagonism was examined by an assay based on measurements of L-glutamate induce...More data for this Ligand-Target Pair
BDBM135949(US8853203, 3 | US8853203, 8 | US9650377, Example 8)
IC50: 585nMAssay Description:Activity of compounds of the present invention was examined by determination to what extent the glutamate-induced elevation of the intracellular calc...More data for this Ligand-Target Pair
BDBM135949(US8853203, 3 | US8853203, 8 | US9650377, Example 8)
BDBM135949(US8853203, 3 | US8853203, 8 | US9650377, Example 8)
IC50: 4.90E+3nMAssay Description:Activity of compounds of the present invention was examined by determination to what extent the glutamate-induced elevation of the intracellular calc...More data for this Ligand-Target Pair
BDBM135949(US8853203, 3 | US8853203, 8 | US9650377, Example 8)
IC50: 4.90E+3nMAssay Description:Activity of compounds of the present invention was examined by determination to what extent the glutamate-induced elevation of the intracellular calc...More data for this Ligand-Target Pair