Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hit in this display   

TargetLeukotriene C4 synthase(Homo sapiens (Human))
Astrazeneca

US Patent

LigandBDBM223259(2-(5-((Cyclopropylmethyl)(4-(trifluoromethyl)napht...)Copy SMILESCopy InChI

Affinity DataIC50:  19nMpH: 7.8Assay Description:In the assay, LTC4 synthase catalyses the reaction where the substrate LTA4 is converted to LTC4. Recombinant human LTC4 synthase is expressed in Pic...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
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