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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetB1 bradykinin receptor(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50309011(CHEMBL598349 | N-(4-((5'-chloro-3,3'-difluoro-2'-(...)
Affinity DataIC50:  0.600nMAssay Description:Antagonist activity at bradykinin B1 receptor in human IMR90 cells pretreated with IL1beta assessed as inhibition of DAKD-induced calcium mobilizatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed