Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 9 hits in this display
BDBM50161620(8-Bromo-7-methoxy-1-methyl-2,3,4,5-tetrahydro-1H-b...)
BDBM50161624((S)-8-Bromo-7-methoxy-1-methyl-2,3,4,5-tetrahydro-...)
EC50: 30nMAssay Description:Effective concentration towards 5-hydroxytryptamine 2C receptors transfected in HEK-293 cells was determined by measuring [3H]-phosphoinositol releas...More data for this Ligand-Target Pair
BDBM50161637((R)-8-Bromo-7-methoxy-1-methyl-2,3,4,5-tetrahydro-...)
BDBM50161637((R)-8-Bromo-7-methoxy-1-methyl-2,3,4,5-tetrahydro-...)
BDBM50161620(8-Bromo-7-methoxy-1-methyl-2,3,4,5-tetrahydro-1H-b...)
EC50: 5nMAssay Description:Effective concentration towards 5-hydroxytryptamine 2A receptors transfected in HEK-293 cells was determined by measuring [3H]-phosphoinositol releas...More data for this Ligand-Target Pair
BDBM50161624((S)-8-Bromo-7-methoxy-1-methyl-2,3,4,5-tetrahydro-...)
EC50: 30nMAssay Description:Effective concentration towards 5-hydroxytryptamine 2B receptors transfected in HEK-293 cells was determined by measuring [3H]-phosphoinositol releas...More data for this Ligand-Target Pair
BDBM50161624((S)-8-Bromo-7-methoxy-1-methyl-2,3,4,5-tetrahydro-...)
EC50: 5nMAssay Description:Effective concentration towards 5-hydroxytryptamine 2A receptors transfected in HEK-293 cells was determined by measuring [3H]-phosphoinositol releas...More data for this Ligand-Target Pair
BDBM50161620(8-Bromo-7-methoxy-1-methyl-2,3,4,5-tetrahydro-1H-b...)
EC50: 80nMAssay Description:Effective concentration towards 5-hydroxytryptamine 2B receptors transfected in HEK-293 cells was determined by measuring [3H]-phosphoinositol releas...More data for this Ligand-Target Pair
BDBM50161637((R)-8-Bromo-7-methoxy-1-methyl-2,3,4,5-tetrahydro-...)
EC50: 220nMAssay Description:Effective concentration towards 5-hydroxytryptamine 2C receptors transfected in HEK-293 cells was determined by measuring [3H]-phosphoinositol releas...More data for this Ligand-Target Pair