Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetAngiopoietin-1 receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304208(CHEMBL595406 | N-(4-(benzo[d]thiazol-2-yl)-2-methy...)
Affinity DataIC50:  38nMAssay Description:Inhibition of TIE2 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304208(CHEMBL595406 | N-(4-(benzo[d]thiazol-2-yl)-2-methy...)
Affinity DataIC50:  250nMAssay Description:Inhibition of VEGFR2 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304208(CHEMBL595406 | N-(4-(benzo[d]thiazol-2-yl)-2-methy...)
Affinity DataIC50:  250nMAssay Description:Inhibition of wild type EGF-R by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304208(CHEMBL595406 | N-(4-(benzo[d]thiazol-2-yl)-2-methy...)
Affinity DataIC50:  340nMAssay Description:Inhibition of VEGFR3 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304208(CHEMBL595406 | N-(4-(benzo[d]thiazol-2-yl)-2-methy...)
Affinity DataIC50:  340nMAssay Description:Inhibition of Aurora-A by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304208(CHEMBL595406 | N-(4-(benzo[d]thiazol-2-yl)-2-methy...)
Affinity DataIC50:  440nMAssay Description:Inhibition of Aurora-B by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304208(CHEMBL595406 | N-(4-(benzo[d]thiazol-2-yl)-2-methy...)
Affinity DataIC50:  490nMAssay Description:Inhibition of ERBB2 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304208(CHEMBL595406 | N-(4-(benzo[d]thiazol-2-yl)-2-methy...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of PDGFRbeta by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed