Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422383(CHEMBL1203235)
Affinity DataIC50:  3.20nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422383(CHEMBL1203235)
Affinity DataIC50:  2.14E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50422383(CHEMBL1203235)
Affinity DataIC50:  4.68E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed