Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 154 hits in this display
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 0.0350nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) incubated for 120 mins by Perkin Elmer electrophoretic mobility shift platform methodMore data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 0.0350nMAssay Description:Inhibition of full length recombinant human GST or His-tagged VEGFR2 using poly (Glu, Tyr) as substrate by AlphaScreen assayMore data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 1.30nMAssay Description:Inhibition of full length recombinant human GST or His-tagged c-Met using poly (Glu, Tyr) as substrate by luciferase coupled chemiluminescence assayMore data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 3.20nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 5.20nMAssay Description:Inhibition of wildtype RET (unknown origin) incubated for 120 mins by Perkin Elmer electrophoretic mobility shift platform methodMore data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 8nMAssay Description:Inhibition of recombinant RET M918T (unknown origin) incubated for 120 mins by Perkin Elmer electrophoretic mobility shift platform methodMore data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 9.90nMpH: 7.4 T: 2°CAssay Description:Briefly, 20 μg/mL poly (Glu,Tyr) 4:1 (Sigma) was pre-coated in 96-well plates as a substrate. A 50 μL aliquot of 10 μmol/L ATP solutio...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 19nMAssay Description:Inhibition of c-MET (unknown origin) using FAM-labelled peptide as substrate measured after 10 mins by mobility shift assayMore data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 20nMAssay Description:Inhibition of TPR-tagged met (unknown origin) expressed in mouse BAF3 cells assessed as inhibition of cell proliferation after 72 hrs by MTT assayMore data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 22nMAssay Description:Inhibition of TPR-tagged met (unknown origin) expressed in mouse BAF3 cells assessed as inhibition of cell proliferation after 72 hrs by MTT assayMore data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 34nMAssay Description:Inhibition of recombinant CCDC6-RET (unknown origin) incubated for 120 mins by Perkin Elmer electrophoretic mobility shift platform methodMore data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 45nMAssay Description:In order to assess the activity of chemical compounds against the relevant kinase of interest, the Caliper LifeSciences electrophoretic mobility shif...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 45nMAssay Description:Inhibition of recombinant RET V804L (unknown origin) incubated for 120 mins by Perkin Elmer electrophoretic mobility shift platform methodMore data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: <50nMAssay Description:Kinase Activity was measured and profiled by EMD Millipore according to the Kinase Profiler Service Assay Protocols Protocol Guide Volume 57. The res...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: <50nMAssay Description:Kinase Activity was measured and profiled by EMD Millipore according to the Kinase Profiler Service Assay Protocols Protocol Guide Volume 57. The res...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: <50nMAssay Description:Kinase Activity was measured and profiled by EMD Millipore according to the Kinase Profiler Service Assay Protocols Protocol Guide Volume 57. The res...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: <50nMAssay Description:Kinase Activity was measured and profiled by EMD Millipore according to the Kinase Profiler Service Assay Protocols Protocol Guide Volume 57. The res...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: <50nMAssay Description:Kinase Activity was measured and profiled by EMD Millipore according to the Kinase Profiler Service Assay Protocols Protocol Guide Volume 57. The res...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 72nMAssay Description:Inhibition of wildtype human TRKA using poly (Glu,Tyr) 4:1 as substrate in presence of [gamma-33P]ATP by hotspot kinase assayMore data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 219nMAssay Description:In each well of a 384-well plate, 7.5 nM-10 nM of wild type RET (ProQinase 1090-0000-1) was incubated in a total of 12.5 μL of buffer (100 mM HE...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 219nMAssay Description:A compound described herein can be tested in vitro for inhibition of wild-type RET and various mutant RET kinases, including e.g., RET V804L, RET V80...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 219nMAssay Description:In order to assess the activity of chemical compounds against the relevant kinase of interest, the Caliper LifeSciences electrophoretic mobility shif...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 585nMAssay Description:In each well of a 384-well plate, 7.5 nM-10 nM of wild type RET (ProQinase 1090-0000-1) was incubated in a total of 12.5 μL of buffer (100 mM HE...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 585nMAssay Description:In each well of a 384-well plate, 7.5 nM-10 nM of mutant RET (ProQinase 1096-0000-1) is incubated in a total of 12.5 μL of buffer (100 mM HEPES ...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
IC50: 585nMAssay Description:In order to assess the activity of chemical compounds against the relevant kinase of interest, the Caliper LifeSciences electrophoretic mobility shif...More data for this Ligand-Target Pair
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
BDBM50021574(BMS-907351 | CABOZANTINIB | CHEBI:72317 | Cabomety...)
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