Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 36 hits in this display
IC50: 56nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: 4.20E+4nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged Aurora kinase-A (1 to 403 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged FAK cytoplasmic domain (376 to 1052 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged YES (1 to 543 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged BRK (2 to 451 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged ABL (2 to 1130 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged RAF1 catalytic domain (306 to 648 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged AKT1 catalytic domain (104 to 480 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged PKCzeta (1 to 592 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged PKCalpha (1 to 351 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged LTK cytoplasmic domain (498 to 796 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged p38-alpha (9 to 352 residues) expressed in Escherichia coli expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KIT cytoplasmic domain (544 to 976 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged EPHA2 cytoplasmic domain (572 to 976 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged INSR cytoplasmic domain (1005 to 1310 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged IGF1R cytoplasmic domain (959 to 1367 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged DDR1 cytoplasmic domain (444 to 876 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged PKCbeta2 (1 to 673 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -pirenzepine providing a measure of muscarinic m1 receptor antagonist affinityMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged FGFR2 cytoplasmic domain (399 to 821 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged AXL cytoplasmic domain (464 to 885 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged RON cytoplasmic domain (979 to 1400 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged MET cytoplasmic domain (956 to 1390 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDR cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:Inhibition of recombinant full length human N-terminal GST-tagged LCK (1 to 509 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
IC50: >5.00E+4nMAssay Description:In vitro 100 nM cortex affinity to displace [3H]- -CD providing a measure of muscarinic m1 receptor agonist affinityMore data for this Ligand-Target Pair