Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetAngiopoietin-1 receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304218(CHEMBL594661 | N-[4-(Benzo[d]thiazol-2''-yl)-2-flu...)
Affinity DataIC50:  360nMAssay Description:Inhibition of TIE2 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304218(CHEMBL594661 | N-[4-(Benzo[d]thiazol-2''-yl)-2-flu...)
Affinity DataIC50:  390nMAssay Description:Inhibition of Aurora-A by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304218(CHEMBL594661 | N-[4-(Benzo[d]thiazol-2''-yl)-2-flu...)
Affinity DataIC50:  410nMAssay Description:Inhibition of Aurora-B by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304218(CHEMBL594661 | N-[4-(Benzo[d]thiazol-2''-yl)-2-flu...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of wild type EGF-R by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304218(CHEMBL594661 | N-[4-(Benzo[d]thiazol-2''-yl)-2-flu...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ERBB2 by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50304218(CHEMBL594661 | N-[4-(Benzo[d]thiazol-2''-yl)-2-flu...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of PDGFRbeta by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed