Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 13 hits in this display
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
IC50: 4.30E+3nMAssay Description:Inhibition of human EGFR expressed in human A431 cells using poly(Glu4/Tyr) and [gamma32P]ATP as substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
IC50: 5.10E+3nMpH: 7.6 T: 2°CAssay Description:The activity of EGFR, preactivated with EGF, is measured by its ability to transfer terminal phosphate from [gamma-32P]ATP to poly(GAT) substrate.More data for this Ligand-Target Pair
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
IC50: 7.00E+3nMAssay Description:Inhibition of recombinant human VEGFR-2 using poly(Glu4/Tyr) and [gamma32P]ATP as substrate after 1 hr by scintillation countingMore data for this Ligand-Target Pair
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
IC50: >1.00E+4nMAssay Description:inhibition of human recombinant CDK5/p25 using histone H1 as substrate by scintillation counting in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)
BDBM3530(6,7-dimethoxy-N-phenylquinazolin-4-amine | CHEMBL5...)