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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

Target5'-nucleotidase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM222262((Z)-4-(2-((E)-4-(3,4-dimethoxyphenyl)-1-morpholino...)
Affinity DataIC50:  260nMpH: 7.4 T: 2°CAssay Description:The ecto-5'-nucleotidase inhibition assay was performed according to our previously reported protocol [Raza et al., Med. Chem., 8:1133-1139]. The com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntestinal-type alkaline phosphatase(Bos taurus (Cattle))
Comsats Institute Of Information Technology

LigandPNGBDBM222262((Z)-4-(2-((E)-4-(3,4-dimethoxyphenyl)-1-morpholino...)
Affinity DataIC50:  350nMpH: 9.8 T: 2°CAssay Description:Alkaline phosphatase assay was optimized and performed in the same way as previously reported method with slight modifications [Sergienko et al., Nat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5'-nucleotidase(Rattus norvegicus (Rat))
Comsats Institute Of Information Technology

LigandPNGBDBM222262((Z)-4-(2-((E)-4-(3,4-dimethoxyphenyl)-1-morpholino...)
Affinity DataIC50:  7.41E+3nMpH: 7.4 T: 2°CAssay Description:The ecto-5'-nucleotidase inhibition assay was performed according to our previously reported protocol [Raza et al., Med. Chem., 8:1133-1139]. The com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed