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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Medical University Of South Carolina

LigandPNGBDBM26632((5Z)-5-[(4-methoxyphenyl)methylidene]-1,3-thiazoli...)
Affinity DataIC50:  300nMAssay Description:The primary screen and evaluation of the compounds was conducted using an ATP-depletion assay. Recombinant human Pim kinase was incubated with S6 kin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Medical University Of South Carolina

LigandPNGBDBM26632((5Z)-5-[(4-methoxyphenyl)methylidene]-1,3-thiazoli...)
Affinity DataIC50:  5.10E+3nMpH: 7.0 T: 2°CAssay Description:The primary screen and evaluation of the compounds was conducted using an ATP-depletion assay. Recombinant human Pim kinase was incubated with S6 kin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM26632((5Z)-5-[(4-methoxyphenyl)methylidene]-1,3-thiazoli...)
Affinity DataIC50:  4.08E+4nMAssay Description:Inhibition of aldose reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed