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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Ariad Gene Therapeutics

Curated by ChEMBL
LigandPNGBDBM50132547(1-Phenylacetyl-piperidine-2-carboxylic acid 1-(3-c...)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibition of binding to Phe36Val (F36V) mutant of FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Ariad Gene Therapeutics

Curated by ChEMBL
LigandPNGBDBM50132547(1-Phenylacetyl-piperidine-2-carboxylic acid 1-(3-c...)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibition of binding to Phe36Val (F36V) mutant of FK506 binding protein 12More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Ariad Gene Therapeutics

Curated by ChEMBL
LigandPNGBDBM50132547(1-Phenylacetyl-piperidine-2-carboxylic acid 1-(3-c...)
Affinity DataIC50:  1.53E+3nMAssay Description:Binding affinity for Mutant F36V-FK506 binding protein by competitive assay based on fluorescence polarization.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed