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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50401375(CHEMBL2205814)
Affinity DataKi:  101nMAssay Description:Displacement of [3H](+)-pentazocine from rat brain sigma1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50401375(CHEMBL2205814)
Affinity DataKi:  1.78E+3nMAssay Description:Binding affinity to Histamine H2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50401375(CHEMBL2205814)
Affinity DataKi:  1.87E+3nMAssay Description:Binding affinity to alpha2C adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50401375(CHEMBL2205814)
Affinity DataKi:  4.27E+3nMAssay Description:Binding affinity to SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50401375(CHEMBL2205814)
Affinity DataKi:  6.87E+3nMAssay Description:Binding affinity to 5-HT7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50401375(CHEMBL2205814)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to alpha1A adrenergicMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50401375(CHEMBL2205814)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5-HT1B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed