Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL

LigandBDBM50129259(CHEMBL3629539)Copy SMILESCopy InChI

Affinity DataKi:  3.55E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells after 2 hrs by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatents

In DepthDetails ArticlePubMed
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TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL

LigandBDBM50129259(CHEMBL3629539)Copy SMILESCopy InChI

Affinity DataKi:  4.30E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells after 2 hrs by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair

Target InfoReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatents

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL

LigandBDBM50129259(CHEMBL3629539)Copy SMILESCopy InChI

Affinity DataKi:  5.40E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells after 2 hrs by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair

Target InfoReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatents

In DepthDetails ArticlePubMed
Copy BDB DOI