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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAminopeptidase N(Sus scrofa (Pig))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50144913(CHEMBL3765067)
Affinity DataIC50:  460nMAssay Description:Inhibition of APN in porcine kidney microsomes preincubated for 5 mins before L-leu-p-nitroanilide substrate addition for 30 mins by plate reader ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase (HDAC1 and HDAC2)(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50144913(CHEMBL3765067)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HDAC1/HDAC2 in human HeLa cells nuclear extract preincubated for 5 mins before Boc-Lys (acetyl)-AMC substrate addition for 30 mins by m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed