Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
BDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
BDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
BDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
BDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
BDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
BDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
BDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
BDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
EC50: 130nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO Flp-In cells assessed as stimulation of acetylcholine-induced ERK1/2 ...More data for this Ligand-Target Pair
BDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
EC50: 680nMAssay Description:Positive allosteric modulation of Gqi5-fused human M4 AChR assessed as increase in acetylcholine-induced calcium mobilizationMore data for this Ligand-Target Pair
BDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)
BDBM48043(3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyrid...)