Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 15 hits in this display
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
IC50: 431nMAssay Description:In a 384 well polypropylene plate, c-FMS (0.14 nM, Carna 08-155) was pre-incubated in a 100 mM Hepes-NaOH pH 7.5 buffer containing 0.01% Triton X-100...More data for this Ligand-Target Pair
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
IC50: 4.37E+3nMAssay Description:In a 384 well polypropylene plate, TrkB (0.6 nM, Carna 08-187) was pre-incubated in a 100 mM Hepes-NaOH pH 7.5 buffer containing 0.01% Triton X-100, ...More data for this Ligand-Target Pair
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
BDBM164921(US10166239, Ex. 3-29 | US11406644, Example 3-29 | ...)
IC50: 8.98E+3nMAssay Description:In a 384 well polypropylene plate, TrkA (0.4 nM, Carna 08-186) was pre-incubated in a 100 mM Hepes-NaOH pH 7.5 buffer containing 0.01% Triton X-100, ...More data for this Ligand-Target Pair