Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50418751(CHEMBL1796032)
Affinity DataKi:  191nMAssay Description:Displacement of [125I]BE-2254 from human adrenergic alpha1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50418751(CHEMBL1796032)
Affinity DataKi:  331nMAssay Description:Displacement of [125I]BE-2254 from human adrenergic Alpha-1B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50418751(CHEMBL1796032)
Affinity DataKi:  389nMAssay Description:Displacement of [125I]BE-2254 from human adrenergic Alpha-1D receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed