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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetAdenosine receptor A1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50025707(5-(2,4-Dimethoxy-phenyl)-1,3-dimethyl-1,6-dihydro-...)
Affinity DataIC50:  5.43E+3nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membrane preparations using N6-[3H]-cyclohexyladenosine as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed