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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Melanin-concentrating hormone receptor 1
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM50340203
(CHEMBL1760249 | N-(3-chlorophenyl)-2-((3R,4S)-4-(4...)
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Affinity Data
IC50: 30nM
Assay Description:
Displacement of [125I]-MCH from MCHR1 after 2 hrs by scintillation counting
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Melanin-concentrating hormone receptor 1
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM50340203
(CHEMBL1760249 | N-(3-chlorophenyl)-2-((3R,4S)-4-(4...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 44nM
Assay Description:
Antagonist activity at MCHR1 by aequorin bioluminescence assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Potassium voltage-gated channel subfamily H member 2
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM50340203
(CHEMBL1760249 | N-(3-chlorophenyl)-2-((3R,4S)-4-(4...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.62E+3nM
Assay Description:
Displacement of [3H]-dofetilide from human ERG expressed in human HEK293 cells after 90 mins by scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
UniProtKB/TrEMBL
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI