Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
The Medicines Company (Leipzig)

US Patent
LigandPNGBDBM104920(US8569313, Inhibitor 35)
Affinity DataKi:  145nMAssay Description:Inhibition assay using matriptase enzymeMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
The Medicines Company (Leipzig)

US Patent
LigandPNGBDBM50254024((+/-)-4'-Methoxy-biphenyl-3-sulfonic acid [2-[4-(2...)
Affinity DataKi:  145nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254024((+/-)-4'-Methoxy-biphenyl-3-sulfonic acid [2-[4-(2...)
Affinity DataKi:  776nMAssay Description:Inhibition of plasmin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254024((+/-)-4'-Methoxy-biphenyl-3-sulfonic acid [2-[4-(2...)
Affinity DataKi:  9.80E+3nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254024((+/-)-4'-Methoxy-biphenyl-3-sulfonic acid [2-[4-(2...)
Affinity DataKi:  5.50E+4nMAssay Description:Inhibition of factor 10a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254024((+/-)-4'-Methoxy-biphenyl-3-sulfonic acid [2-[4-(2...)
Affinity DataKi:  1.29E+5nMAssay Description:Inhibition of uPA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed