Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
BDBM50086128(2-(4-Methoxy-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]q...)
Ki: 16nMAssay Description:Binding affinity towards human adenosine A3 receptor expressed in HEK-293 cells in presence of [125I]-AB-MECA at a concentration of 1 uMMore data for this Ligand-Target Pair
BDBM50086128(2-(4-Methoxy-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]q...)
BDBM50086128(2-(4-Methoxy-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]q...)
BDBM50086128(2-(4-Methoxy-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]q...)
Ki: 934nMAssay Description:Binding affinity towards adenosine A1 receptor of bovine brain membrane in presence of [3H]-CHA at a concentration of 20 uMMore data for this Ligand-Target Pair
BDBM50086128(2-(4-Methoxy-phenyl)-2H,5H-[1,2,4]triazolo[4,3-a]q...)