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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50024377(CHEMBL2113037)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of [125I]-NDP- alpha-MSH binding to human melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50024377(CHEMBL2113037)
Affinity DataIC50:  26nMAssay Description:Inhibition of [125I]-NDP- alpha-MSH binding to human melanocortin 4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50024377(CHEMBL2113037)
Affinity DataIC50:  230nMAssay Description:Inhibition of [125I]-NDP- alpha-MSH binding to human melanocortin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50024377(CHEMBL2113037)
Affinity DataIC50:  420nMAssay Description:Inhibition of [125I]-NDP- alpha-MSH binding to human melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50024377(CHEMBL2113037)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of [125I]-NDP- alpha-MSH binding to human melanocortin 5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50024377(CHEMBL2113037)
Affinity DataEC50:  390nMAssay Description:Effective concentration at human melanocortin 4 receptor in cAMP release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50024377(CHEMBL2113037)
Affinity DataEC50:  2.40E+3nMAssay Description:Effective concentration against human melanocortin 5 receptor in cAMP release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed