Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetStromelysin-1(Homo sapiens (Human))
Hokkaido Collaboration Center

Curated by ChEMBL
LigandPNGBDBM50131384((2R,3S,4S,5S)-3,4,5-Trihydroxy-1-(4-methoxy-benzen...)
Affinity DataKi:  490nMAssay Description:Inhibition of recombinant human matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Hokkaido Collaboration Center

Curated by ChEMBL
LigandPNGBDBM50131384((2R,3S,4S,5S)-3,4,5-Trihydroxy-1-(4-methoxy-benzen...)
Affinity DataKi:  510nMAssay Description:Inhibition of recombinant human TNF-alpha converting enzyme (TACE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Hokkaido Collaboration Center

Curated by ChEMBL
LigandPNGBDBM50131384((2R,3S,4S,5S)-3,4,5-Trihydroxy-1-(4-methoxy-benzen...)
Affinity DataKi:  780nMAssay Description:Inhibition of recombinant human matrix metalloproteinase-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Hokkaido Collaboration Center

Curated by ChEMBL
LigandPNGBDBM50131384((2R,3S,4S,5S)-3,4,5-Trihydroxy-1-(4-methoxy-benzen...)
Affinity DataKi: >850nMAssay Description:Inhibition of recombinant human matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed