Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetNeutrophil collagenase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50077420((R)-5-(4-Methoxy-benzenesulfonyl)-1-methyl-4,5,6,7...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration against human matrix metalloproteinase-8 (human neutrophil collagenase, MMP-8)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50077420((R)-5-(4-Methoxy-benzenesulfonyl)-1-methyl-4,5,6,7...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human neutrophil collagenase [Matrix Metalloprotease-8, MMP-8]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50077420((R)-5-(4-Methoxy-benzenesulfonyl)-1-methyl-4,5,6,7...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration of the compound against human matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed