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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of matrix metalloproteinase-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataIC50:  1.30nMAssay Description:Phosphodiesterase 4 inhibitory activity measured against guinea pig macrophage homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against recombinant matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against recombinant matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed