Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50129450((S)-1-(9H-Carbazol-4-yloxy)-3-[1-(3,4-dimethoxy-be...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonistic activity against cloned human beta1-AR (beta2-adrenergic receptor) in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50129450((S)-1-(9H-Carbazol-4-yloxy)-3-[1-(3,4-dimethoxy-be...)
Affinity DataEC50:  20nMAssay Description:Agonistic activity against cloned human beta3-AR (beta3-adrenergic receptor) in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50129450((S)-1-(9H-Carbazol-4-yloxy)-3-[1-(3,4-dimethoxy-be...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonistic activity against cloned human beta1-AR (beta1-adrenergic receptor) in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed