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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human))
Rhone-Poulenc Rorer
Curated by
ChEMBL
Ligand
BDBM50090352
(3-(3-Cyclopentyloxy-4-methoxy-benzenesulfonyl)-7-p...)
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Affinity Data
IC50: 6.90nM
Assay Description:
Phosphodiesterase 4 inhibitory activity measured against guinea pig macrophage homogenate
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Interstitial collagenase
(Homo sapiens (Human))
Rhone-Poulenc Rorer
Curated by
ChEMBL
Ligand
BDBM50090352
(3-(3-Cyclopentyloxy-4-methoxy-benzenesulfonyl)-7-p...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of Matrix metalloproteinase-1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Stromelysin-1
(Homo sapiens (Human))
Rhone-Poulenc Rorer
Curated by
ChEMBL
Ligand
BDBM50090352
(3-(3-Cyclopentyloxy-4-methoxy-benzenesulfonyl)-7-p...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibitory activity against recombinant matrix metalloproteinase-3
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
72 kDa type IV collagenase
(Homo sapiens (Human))
Rhone-Poulenc Rorer
Curated by
ChEMBL
Ligand
BDBM50090352
(3-(3-Cyclopentyloxy-4-methoxy-benzenesulfonyl)-7-p...)
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Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibitory activity against recombinant matrix metalloproteinase-2
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI