Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50090352(3-(3-Cyclopentyloxy-4-methoxy-benzenesulfonyl)-7-p...)
Affinity DataIC50:  6.90nMAssay Description:Phosphodiesterase 4 inhibitory activity measured against guinea pig macrophage homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50090352(3-(3-Cyclopentyloxy-4-methoxy-benzenesulfonyl)-7-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50090352(3-(3-Cyclopentyloxy-4-methoxy-benzenesulfonyl)-7-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against recombinant matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50090352(3-(3-Cyclopentyloxy-4-methoxy-benzenesulfonyl)-7-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against recombinant matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed