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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University Of Tokyo

LigandPNGBDBM23846(5,25-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1...)
Affinity DataIC50:  2.50E+4nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-glucosidase MAL32(Saccharomyces cerevisiae)
University Of Tokyo

LigandPNGBDBM23846(5,25-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1...)
Affinity DataIC50: >3.00E+4nMpH: 7.0 T: 2°CAssay Description:The alpha-glucosidase inhibitory activity of test compounds was determined in a 96-well plate format. The reaction mixture containing enzyme and chro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
University Of Tokyo

LigandPNGBDBM23846(5,25-dimethoxy-14-oxapentacyclo[20.2.2.2^{10,13}.1...)
Affinity DataIC50:  4.60E+4nMAssay Description:Human embryonic kidney (HEK) 293 cells were cultured in D-MEM medium. Transfections were performed by the calcium phosphate coprecipitation method. T...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed