Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetKinesin-like protein KIF20A(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50140929(CHEMBL3754608)
Affinity DataIC50:  230nMAssay Description:Inhibition of microtubule-stimulated N-terminal MKLP-2 (56 to 505 residues) ATPase activity isolated from human hepatocellular carcinoma cells by pyr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF20A(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50140929(CHEMBL3754608)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of N-terminal MKLP2 (56 to 505 residues) ATPase basal activity isolated from human hepatocellular carcinoma cells by pyruvate kinase/lacta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50140929(CHEMBL3754608)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50140929(CHEMBL3754608)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate after 30 mins in presence of [gamma-33 P] ATP by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed