Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelatonin receptor(RABBIT)
Northwestern University

Curated by PDSP Ki Database
LigandPNGBDBM85053(1-[2-(5-Methoxy-1H-indol-3-yl)ethyl]pyrrolidin-2-o...)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Northwestern University

Curated by PDSP Ki Database
LigandPNGBDBM85053(1-[2-(5-Methoxy-1H-indol-3-yl)ethyl]pyrrolidin-2-o...)
Affinity DataKi:  18.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor(RABBIT)
Northwestern University

Curated by PDSP Ki Database
LigandPNGBDBM85053(1-[2-(5-Methoxy-1H-indol-3-yl)ethyl]pyrrolidin-2-o...)
Affinity DataKi:  58nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Northwestern University

Curated by PDSP Ki Database
LigandPNGBDBM85053(1-[2-(5-Methoxy-1H-indol-3-yl)ethyl]pyrrolidin-2-o...)
Affinity DataKi:  289nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed