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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Melatonin receptor type 1A/1B
(Homo sapiens (Human))
University Of Urbino
Curated by
ChEMBL
Ligand
BDBM50230659
(CHEMBL37549)
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Affinity Data
Ki: 2.20nM
Assay Description:
Inhibition of 2-[125I]iodomelatonin binding to melatonin receptor in quail brain as 1/Ka
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
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Article
PubMed
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Target
Melatonin receptor type 1C
(Gallus gallus)
Universit£
Curated by
ChEMBL
Ligand
BDBM50230659
(CHEMBL37549)
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Affinity Data
Ki: 2.5nM
Assay Description:
Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligand
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melatonin receptor type 1A/1B
(Homo sapiens (Human))
University Of Urbino
Curated by
ChEMBL
Ligand
BDBM50230659
(CHEMBL37549)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.0000500nM
Assay Description:
Monophasic inhibitory concentration against melatonin receptor was measured on ovine pars tuberalis membrane.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melatonin receptor type 1A/1B
(Homo sapiens (Human))
University Of Urbino
Curated by
ChEMBL
Ligand
BDBM50230659
(CHEMBL37549)
Copy SMILES
Copy InChI
Affinity Data
Kd: 0.000453nM
Assay Description:
Binding affinity to melatonin receptor measured on ovine pars tuberalis membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI