Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMelatonin receptor type 1B(Homo sapiens (Human))
Iqm-Csic

Curated by ChEMBL
LigandPNGBDBM50096967(CHEMBL3580916)
Affinity DataKi:  190nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-2 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Iqm-Csic

Curated by ChEMBL
LigandPNGBDBM50096967(CHEMBL3580916)
Affinity DataKi:  709nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human melatonin receptor-1 transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Iqm-Csic

Curated by ChEMBL
LigandPNGBDBM50096967(CHEMBL3580916)
Affinity DataEC50:  881nMAssay Description:Agonist activity at human melatonin receptor-2 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Iqm-Csic

Curated by ChEMBL
LigandPNGBDBM50096967(CHEMBL3580916)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human recombinant melatonin receptor-2 expressed in CHO cells assessed as decrease of cAMP level after 10 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Iqm-Csic

Curated by ChEMBL
LigandPNGBDBM50096967(CHEMBL3580916)
Affinity DataEC50:  961nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed