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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Mu-type opioid receptor
(Homo sapiens (Human))
University Of Bath
Curated by
ChEMBL
Ligand
BDBM50249016
(CHEMBL471543 | N-Cyclopropylmethyl-14beta-4'-methy...)
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Affinity Data
Ki: 4.20nM
Assay Description:
Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Kappa-type opioid receptor
(Homo sapiens (Human))
University Of Bath
Curated by
ChEMBL
Ligand
BDBM50249016
(CHEMBL471543 | N-Cyclopropylmethyl-14beta-4'-methy...)
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Copy InChI
Affinity Data
Ki: 36nM
Assay Description:
Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(Homo sapiens (Human))
University Of Bath
Curated by
ChEMBL
Ligand
BDBM50249016
(CHEMBL471543 | N-Cyclopropylmethyl-14beta-4'-methy...)
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Affinity Data
Ki: 270nM
Assay Description:
Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Homo sapiens (Human))
University Of Bath
Curated by
ChEMBL
Ligand
BDBM50249016
(CHEMBL471543 | N-Cyclopropylmethyl-14beta-4'-methy...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 157nM
Assay Description:
Agonist activity at human kappa opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI