Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105773(17-(2-methylallyl)-substituted noroxymorphone deri...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]DADLE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105773(17-(2-methylallyl)-substituted noroxymorphone deri...)
Affinity DataKi: >6.00E+3nMAssay Description:Displacement of [3H]DAMGO from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105773(17-(2-methylallyl)-substituted noroxymorphone deri...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]U-69593 from Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed