Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179286((+)-(S)-1-(3-(6-methoxynaphthalen-1-yl)propyl)-2-m...)
Affinity DataKi:  7.05nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Cavia porcellus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50179286((+)-(S)-1-(3-(6-methoxynaphthalen-1-yl)propyl)-2-m...)
Affinity DataKi:  46.5nMAssay Description:Displacement of [3H](+/-)-emopamil from delta8-delta7 sterol isomerase (SI) site in guinea pig liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed