Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM50427626(CHEMBL2323481 | US9346803, Table 2, Compound 5: 2-...)
BDBM50427626(CHEMBL2323481 | US9346803, Table 2, Compound 5: 2-...)
IC50: 81nMAssay Description:Inhibitors were initially screened for an ability to block the NADP+ dependent oxidation of the artificial substrate S-tetralol catalyzed by AKR1C3. ...More data for this Ligand-Target Pair
BDBM50427626(CHEMBL2323481 | US9346803, Table 2, Compound 5: 2-...)
IC50: >100nMAssay Description:Inhibitors were initially screened for an ability to block the NADP+ dependent oxidation of the artificial substrate S-tetralol catalyzed by AKR1C3. ...More data for this Ligand-Target Pair
BDBM50427626(CHEMBL2323481 | US9346803, Table 2, Compound 5: 2-...)
IC50: >100nMAssay Description:Inhibitors were initially screened for an ability to block the NADP+ dependent oxidation of the artificial substrate S-tetralol catalyzed by AKR1C3. ...More data for this Ligand-Target Pair
BDBM50427626(CHEMBL2323481 | US9346803, Table 2, Compound 5: 2-...)
BDBM50427626(CHEMBL2323481 | US9346803, Table 2, Compound 5: 2-...)
BDBM50427626(CHEMBL2323481 | US9346803, Table 2, Compound 5: 2-...)
BDBM50427626(CHEMBL2323481 | US9346803, Table 2, Compound 5: 2-...)