Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206175(1-(3-methoxybenzyl)-6-methoxy-2,3,4,9-tetrahydro-1...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206175(1-(3-methoxybenzyl)-6-methoxy-2,3,4,9-tetrahydro-1...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50206175(1-(3-methoxybenzyl)-6-methoxy-2,3,4,9-tetrahydro-1...)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of [3H]N-methylscopolamine from muscarinic M4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed