Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50183343(CHEMBL3818506)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [125I]-apelin13 from human APJ receptor expressed in CHOK1 cell membranes after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50183343(CHEMBL3818506)
Affinity DataEC50:  9.90E+3nMAssay Description:Agonist activity at human APJ receptor expressed in cells c-expressing Galphaq16 assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 2(Rattus norvegicus)
Rti International

Curated by ChEMBL
LigandPNGBDBM50183343(CHEMBL3818506)
Affinity DataEC50:  345nMAssay Description:Partial agonist activity at rat NTS2 receptor expressed in CHOK1 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed