Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM270165((2S,3R)N-(5-(5-bromopyridin-3-yl)-4-(2,6-dim...)
BDBM270265(Preparation (2S,3R)N-(5-(5-cyano-3-pyridinyl...)
EC50: 70nMpH: 7.5Assay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...More data for this Ligand-Target Pair
BDBM270165((2S,3R)N-(5-(5-bromopyridin-3-yl)-4-(2,6-dim...)
BDBM270165((2S,3R)N-(5-(5-bromopyridin-3-yl)-4-(2,6-dim...)
BDBM270165((2S,3R)N-(5-(5-bromopyridin-3-yl)-4-(2,6-dim...)
EC50: 2nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair
BDBM270165((2S,3R)N-(5-(5-bromopyridin-3-yl)-4-(2,6-dim...)
EC50: 0.420nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
BDBM270165((2S,3R)N-(5-(5-bromopyridin-3-yl)-4-(2,6-dim...)
EC50: 2nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
BDBM270165((2S,3R)N-(5-(5-bromopyridin-3-yl)-4-(2,6-dim...)
EC50: 0.420nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair